In the noon of October 19, 2016, a teleconference was held to discuss the latest research progresses made in the international collaboration project on GPCRs. Present in the iHuman Institute, ShanghaiTech University, were Professor Ming-Wei Wang (Dean, School of Pharmacy, Fudan University and Director, the National Center for Drug Screening), Drs. Zhijie Liu (Professor and Deputy Director), Gaojie Song (Research Associate Professor) and Suwen Zhao (Research Associate Professor) from the iHuman Institute, Drs. Beili Wu (Professor) and Dehua Yang (Associate Professor) from Shanghai Institute of Materia Medica, Chinese Academy of Sciences as well as Associate Professor Li Ye from School of Pharmacy, Fudan University. Dr. Raymond Stevens (Professor and Director, iHuman Institute and International Adjunct Professor of Fudan School of Pharmacy), Michael Hanson (Director, International GPCR Consortium) and Chris de Graff (Associate Professor, VU University Amsterdam) participated in the discussion via telephone from U.S.A. and the Netherlands, respectively. The attendants reached an agreement as to the near-term priorities and associated action items.