In the morning of October 12, 2016, Dr. Raymond Stevens (Professor of iHuman Institute, ShanghaiTech University and International Adjunct Professor of Fudan School of Pharmacy), Dr. Beili Wu (Professor of Shanghai Institute of Materia Medica, Chinese Academy of Sciences) and Professor Ming-Wei Wang (Dean, School of Pharmacy, Fudan University and Director, the National Center for Drug Screening) met at School of Pharmacy, Fudan University to discuss recent progresses made in the international collaboration program on GPCR. They agreed on the near-term priorities and associated action items. Senior members of the research teams, i.e., Drs. Michael Hanson (joined from U.S.A.), Qiang Zhao, Chris de Graff (joined from the Netherlands), Gaojie Song, Dehua Yang as well as two graduate students, Haonan Zhang and Anna Qiao, participated in this telephone conference.